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IPhepase enzyme enzyme Qalabka Cancelinta Cilmi-baarista (IC50), microsomes beerka aadanaha, lab

Sharraxaadda Gaaban:

Cyp1, Cyp2 iyo qoysaska Cyp2 iyo CYP3 waa Eyzymes-ka ugu weyn ee Cym450 ee ku lug leh dheef-shiid kiimikaad daroogada. Inhibitory effect of drug candidates on seven CYP subtypes, namely CYP1A2, CYP2A6, CYP2C9, CYP2C19, CYP2D6, CYP2E1 and CYP3A4, are commonly investigated by measuring IC50 using selective probe substrates.

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Calaamadaha wax soo saarka

  • Dhex qori

    Microsome - Substrate - Nidaamka dib-u-cusboonaysiinta Nadph - 0.1m PBS (Ph7.4)

    • Qeybta:
      Xirmooyinka dheef-shiid kiimikaadka vitro
    • Shayga no.:
      0115A1.11
    • Cabbirka Unugga:
      0.2ml * 100 tijaabo
    • Unugyada:
      Beer
    • Noocyada:
      Insaan ah
    • Galmo:
      Labood ah
    • Xaaladaha kaydinta iyo gaadiidka:
      Kaydso AT - 70 ° C. Baraf qalalan ayaa la keenay.
    • Nooca Assay:
      Qalabka xakamaynta ee enzyMyme (IC50)
    • Nidaamka Imtixaanka:
      Jutrosto
    • Baaxadda Codsiga:
      Dheecaannada dheef-shiidka daroogada ee vitro

  • Hore:
  • Xiga:
  • Xulashada Luqadda