Nga tuhinga hangarau
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Sulfotransferase (He he) mo te rangahau DDI, te pumau, me te aukati i te waikawa
Nga Kupu matua: Te tarukino - Te Tauhokohoko tarukino (DDI), Sultzotransfitionase (Sultzainsfation, Sultzolic Sultzation, tangata Sult1A3, Sultz1Panui Panui -
CarboxylesAserases (CES) I te konutai tarukino: Te Taha Reachoping me DDI
Kupu matua: Te raau taero - Tauhokohoko tarukino (DDI), Carboxylesterase 1, CarboxylestesAte 2, Ces1, Ces2, Ces2, CestHabolic Haumaru, TauhouPanui Panui -
Tono o Cytochrome P450 (Cyp450) me UDP - Glucuronosyltfenfenfenfe (UGT) INCHAMES I TE WHAKAMAHI - NGĀ TOHUTOHU I TE WHAKAMAHI I TE WHAKAMAHI I TE WHAKAMAHI I TE WHAKAMAHI I TE WHAKAMAHI I TE WHAKAMAHI I TE WHAKAMAHI I TE WHAKAMAHI I TE WHAKAMAHI I TE WHAKAMAHI I TE WHAKAMAHI
Nga kupu matua: Te raau taero - Tauhokohoko tarukino (DDI), Cyp450 (Cyp450 Haumaru, Cyp2B6, Cyp2C8, Cyp2C9Panui Panui -
Te Tangata Tangata me te kararehe kararehe o te whariki koiora mo te whanaketanga tikanga bionantalytical me te Whakamana Tikanga Tikanga
1 Iphase SucturesPridict Vaypecintifechachachachachachasy tangata Bile2Mliphase Monkey Cynomolgus / Macaca Ficticularis Bile, Kaitautoko kotahi, ko te kaituku kotahi, macaca fickuPanui Panui -
Whakawhitihia nga Tiwhikete Uru Cerabrospinal (Tātaritanga CSF) me te Whakawhanake Matrix Hangarau: Te whakaoti i nga konutai hangarau matua i te CNS tarukino Bioanalysis CNS
1 Iphase HuatureSptRoDuctspeCinifyipHalintifeCinifyeKo te tangata Cenomolgus CyNomolgus / Macaca fiebrospinal rere, te tanupene1mliphahaPanui Panui -
5α 5α - AKO TE WHAKAMAHI KAUPAPA: Srd_A1 & Srd_A2 mo te mana sebum i roto i te Pūtaiao Hinengaro
Kupu matua: Momo 1 5α - Momo 2 5α 12 5α - Srd_A1, Srd_A1, Srdwa2, Mahi Adjectoestosterne (DHT) .iphPanui Panui -
Te hautanga o te kiore S9 o te kiore S9: he punaha whakahohenga metabolic mo te vitro genotoxicity me nga whakamatautau moroiti
Kupu matua: OECD 471, OECD 473, OECD 476, OECD 487, Ko te Whakatuturutanga, Te Ope Taonga, Iti Atu, Mini Ahumoana, MicrouclesPanui Panui -
Plasma pūmua herea Dynamics: dialilibrium dialysis me nga tikanga ultrafilting me te tono i DDIS
Kupu matua: He rite ki te dialifrium, ultrafiltration, plasma pūmua herea (ppb), te taapiri o te plap sallsa plasma (pppp), te reanga dialilibrium dialyissisPanui Panui -
Hepatocytes i roto i te metabolism tarukino me te tuku i te tarukino Sirna: te aro mātai i nga punaha tauira puta noa i nga momo
Huarahi Ingoa Huarahi Tuatahi Hepatocesstes Iphase Whakapau Hepatolytes4 - 6millolipiphase Te Moana Takawaenga (Cynomolgus) hepatolycytes, tane5mlillionPanui Panui -
Ko nga Microsomes i roto i te pumau pumau ka tutuki: mahi i roto i te waahanga me te metabolism me te kotabolism ii
Impsomence Iphasencessessciences sigsonspriverseriver a MicrosomeSiphase Microsesiphase ExerSomhas, whakaranu ira tangata, 20MG / Mliphase Monkey (Cynomolgus) Microshos, TanePanui Panui -
Splenocytes i roto i te Rangahau Immonological: puta noa i nga momo me te wehe, te aukati, nga hikoinga tapawha
Kupu matua: Splenocytes (Spls); Cynomolgus Monkey Splenocytes; Rhesus makimaki makimaki splenocytes; Ko te Splenocytes kuri; Cannonocytes; Kiore splenocytes; Ko nga kiore o te kiore; Ko nga tohu Mice Splenocytes; Rapeti Splenocytes; SpPanui Panui -
Te ahunga whakamua i roto i te biohanalysis: Te mahi a LC - MS / MS i te whanaketanga tarukino ophthallic me te whakatipuranga me te nui me te nui o nga rangahau ngawari
Iphase progensprdifireductiphase tangata waiamu quiserf1mliphase monkey (cynomolgus) waimoana wai waikore, ma te kowhatu1Panui Panui