Technical Notes
-
Sulfotransferase(SULT) for DDI Research, Metabolic Stability, and Enzyme Inhibition
Key words: drug-drug interaction (DDI), sulfotransferase (SULT), enzyme inhibition, SULT metabolic, metabolic stability, human SULT1A1 enzyme, human SULT1A3 enzyme, human SULT1B1 enzyme, human SULT1C2Read more -
Carboxylesterases (CES) in Drug Metabolism: Reaction Phenotyping and DDI
Keywords: Drug-Drug Interaction(DDI), Carboxylesterase 1, Carboxylesterase 2, CES1, CES2, Liver Carboxylesterase, Intestinal Carboxylesterase, CES Enzyme Inhibition, Drug Metabolic Stability, ReactionRead more -
Application of Cytochrome p450 (CYP450) and UDP-glucuronosyltransferase (UGT) Enzymes in Drug-drug Interaction Studies Regarding Metabolic Phenotype and Enzyme Inhibition
Key words: drug-drug interaction (DDI), cytochrome p450 (CYP450 enzyme), udp-glucuronosyltransferase (UGT), Enzyme inhibition, CYP450 enzyme metabolic phenotyping study, CYP1A2, CYP2B6, CYP2C8, CYP2C9Read more -
Human & Animal Bile of Blank Biological Matrix for Bioanalytical Method Development and Bioanalytical Method Validation
1 IPHASE Products Product Name Specification IPHASE Human Bile 2mL IPHASE Monkey Cynomolgus/Macaca Fascicularis Bile,Single Donor,Male 2mL IPHASE Monkey Cynomolgus/Macaca FascicuRead more -
Cross Species Cerebrospinal Fluid Analysis (CSF Analysis) and Artificial Matrix Development: Solving Key Technical Bottlenecks in CNS Drug Bioanalysis
1 IPHASE Products Product Specification IPHASE Human Cerebrospinal Fluid 1mL IPHASE Monkey Cynomolgus/Macaca Fascicularis Cerebrospinal Fluid,Male 1mL IPHASE Monkey(Rhesus) CerebRead more -
5α-Reductase Activity Study: SRD5A1 & SRD5A2 for Sebum Control in Cosmetic Science
Keywords: Type 1 5α-Reductase, Type 2 5α-Reductase, 5αR1, 5αR2, SRD5A1, SRD5A2, NADPH, 5α-Reductase Activity, 5α-Reductase Inhibition, Dihydrotestosterone(DHT). IPHRead more -
Induced Rat Liver S9 Fraction: A Metabolic Activation System for In Vitro Genotoxicity and Mutation Tests
Keywords: OECD 471, OECD 473, OECD 476, OECD 487, Mutation Test, Genotoxicity, Genetic Toxicity, Induced Rat Liver S9, Ames Test, Mini Ames Test, Chromosomal Aberration, Micronucleus, HPRT/HGPRT AssayRead more -
Plasma Protein Binding Dynamics: Equilibrium dialysis and Ultrafiltration Methods and Application in DDIs
Keywords: Equilibrium Dialysis, Ultrafiltration, Plasma Protein Binding(PPB), Binding rate of plasma protein(BRPP), Equilibrium Dialysis Device, Equilibrium Dialysis Membrane, Rapid Equilibrium DialysRead more -
Hepatocytes in Drug Metabolism and siRNA Drug Delivery: Evaluating Model Systems Across Species
Product Name Specification Suspension Primary Hepatocytes IPHASE Suspension Human Primary Hepatocytes 4-6million IPHASE Suspension Monkey(Cynomolgus) Hepatocytes,Male 5millionRead more -
Microsomes in Metabolic Stability Assays: Role in Phase I Metabolism and Phase II Metabolism
IPHASE Biosciences Products Product Name Specification Liver Microsomes IPHASE Human Liver Microsomes,Mixed Gender 0.5mL,20mg/mL IPHASE Monkey(Cynomolgus) Liver Microsomes,MaleRead more -
Splenocytes in Immunological Research: Across Species and Isolation, Freezing, Thawing Steps
Keywords: Splenocytes(SPLs); Cynomolgus Monkey Splenocytes; Rhesus Monkey Splenocytes; Dog Splenocytes; Canine Splenocytes; Rat Splenocytes; Mouse Splenocytes; Mice Splenocytes; Rabbit Splenocytes; SpRead more -
Advancements in Bioanalysis: The Role of LC-MS/MS in Ophthalmic Drug Development and Aqueous and Vitreous Humor Studies
IPHASE Products Product Name Specification IPHASE Human Aqueous Fluid 1mL IPHASE Monkey(Cynomolgus) Aqueous Fluid,Male 1mL IPHASE Rabbit(New Zealand White) Aqueous Fluid,Male 1Read more