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IPHASE Phase II Metabolic Stability Kit, Rat(Sprague-Dawley)

ʻO ka wehewehe pōkole:

ʻO ka Phase II metabolism, i ʻike ʻia ʻo ka hoʻopaʻa paʻa ʻana, e pili ana i ka hopena i hui pū ʻia nā metabolites a i ʻole nā ​​​​lāʻau prototype me nā molekele liʻiliʻi endogenous ma o nā enzymes phase II, e alakaʻi ana i ka hōʻemi ʻana o ka ʻona, ka hana, a i ʻole ka polarity o nā prodrugs. I ka hana II metabolism, ʻo ka hopena maʻamau ka glucuronidation, kahi i hoʻopaʻa ʻia ai ka uridine diphosphate glucuronic acid (UDPGA) i ka prodrug ma o ka catalyzation e glucuronyl transferase i nā microsomes. Hoʻonui ka glucuronide i ka wai-solubility o nā metabolites e hoʻonui i ka excretion. Hiki ke kūkulu hou ʻia ka ʻōnaehana metabolic phase II e ka hui pū ʻana o nā microsomes ate a me UGT a hoʻohana ʻia e aʻo i ka pae II metabolic stability o nā moho lāʻau i vitro.

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Huahana Huahana

  • wehewehe huahana

    Microsome|Substrate| UGT Incubation System| 0.1M PBS (pH7.4)

    • Māhele:
      In vitro metabolism kits
    • 'ikamu NO.:
      0112D1.02
    • Lahi Unit:
      0.2mL*50 hoao
    • Tissue:
      ʻāpaʻa
    • ʻano:
      Iole
    • Moe:
      Wahine
    • Nā kūlana mālama a me ka lawe ʻana:
      E kūʻai ma -70°C. Hāʻawi ʻia ka hau maloʻo.
    • ʻAno hoʻāʻo:
      Māhele II ʻOihana Hoʻokūpaʻa Metabolic (UGT)
    • Pūnaehana hoʻāʻo:
      Microsome
    • Ka laulā o ka noi:
      In vitro Assessment of Metabolic Stability

  • Mua:
  • Aʻe:
  • Koho ʻŌlelo