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IPHASE Phase II Metabolic Stability Kit,Gonzo(Sprague-Dawley)

Tsanangudzo Pfupi

Phase II metabolism, inozivikanwawo seyekusunga maitiro, inoreva maitiro umo chikamu I metabolites kana prototype zvinodhaka zvinosanganiswa ne endogenous mamorekuru madiki kuburikidza nechikamu II ma enzymes, zvichikonzera kudzikiswa kwehupfu, chiitiko, kana polarity yezvigadzirwa. Muchikamu chechipiri chemetabolism, chinowanzoitika ndeye glucuronidation, panguva iyo uridine diphosphate glucuronic acid (UDPGA) inosungirirwa kune prodrug kuburikidza necatalyzation neglucuronyl transferase muma microsomes. Iyo glucuronide yakaumbwa inowedzera mvura - kunyungudika kwematabolites kuwedzera kubuda. Iyo phase II metabolic system inogona kuvakwazve nekusanganiswa kwechiropa microsomes uye UGT uye inoshandiswa kudzidza chikamu chechipiri metabolic kugadzikana kwevanoda zvinodhaka mu vitro.

Product Detail

Product Tags

  • Product discription

    Microsome|Substrate| UGT Incubation System| 0.1M PBS (pH7.4)

    • Category:
      In vitro metabolism kits
    • Chinhu NO.:
      0112D1.02
    • Saizi yeyuniti:
      0.2mL * 50 bvunzo
    • Chirwere:
      Chiropa
    • Mhando:
      Rat
    • Bonde:
      Mukadzi
    • Mamiriro ekuchengetedza uye chekufambisa:
      Chengetedza pa -70°C. Aizi yakaoma inounzwa.
    • Assay Type:
      Phase II Metabolic Stability Kit (UGTs)
    • Test System:
      Microsome
    • Kuwanda kwekushandisa:
      In vitro Ongororo yeMetabolic Kugadzikana

  • Zvakapfuura:
  • Zvinotevera:
  • Kusarudza Mutauro