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Ipase Enzyme inhibition Kev Tshawb Fawb Cov Khoom Siv (IC50), tib neeg lub siab microsomost, poj niam

Cov lus piav qhia luv luv:

CYP1, CYP2 thiab CYP3 tsev neeg yog qhov tseem ceeb CY450 enzymes koom nrog tshuaj metabolism. Inhibitory effect of drug candidates on seven CYP subtypes, namely CYP1A2, CYP2A6, CYP2C9, CYP2C19, CYP2D6, CYP2E1 and CYP3A4, are commonly investigated by measuring IC50 using selective probe substrates.

Khoom Qhia Qhia

Khoom Ntawv

  • Cov Khoom Nrhabrraption discription

    Microsome - Substrate - Nadph Kev Txhim Kho Txheej Txheem - 0.1m PBS (Ph7.4

    • Qeb:
      Hauv cov khoom siv vitro metabolism
    • Yam khoom tsis tau.:
      0115a1.12
    • Chav Tsev Loj:
      0.2ml * 100 xeem
    • Cov ntaub so ntswg:
      Nplooj siab
    • Hom:
      Tus neeg
    • Sib deev:
      Tus pojniam
    • Kev Cia Cov Neeg Cia thiab Tsheb Thauj Mus Los:
      Khw ntawm - 70 ° C. Dej khov kom qhuav.
    • Yam tshuaj uas:
      Enzyme Inhibition Khoom (IC50)
    • Kuaj System:
      Microstre
    • Cov tau txais daim ntawv thov:
      Hauv VeneRo Tshuaj Tshuaj Yeeb Yam

  • Yav dhau los:
  • Tom ntej:
  • Lus Xaiv