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Iphase Ntu II metabolic Stability Cov Khoom Siv, Monkey (Cynomolgus)

Cov lus piav qhia luv luv:

Theem II metabolism, tseem hu ua cov tshuaj tiv thaiv kab mob, hais txog cov tshuaj tiv thaiv me me, ua haujlwm, lossis polarity ntawm produgs. Nyob rau hauv theem II metabolism, feem ntau cov tshuaj tiv thaiv yog gluidine diphosphate looj suab paj nruag los ntawm kev hloov pauv ntawm cov microsomes. Lub glucuronide tsim cov dej nce ntxiv - solubility ntawm metabolites los txhim kho lub excretion. Cov theem II metabolic system tuaj yeem tsim kho dua los ntawm kev sib xyaw ntawm daim tawv nqaij microsomes thiab siv los kawm theem II metabolic stability ntawm cov neeg sib tw ntawm cov tshuaj sib tw hauv vitro.

Khoom Qhia Qhia

Khoom Ntawv

  • Cov Khoom Nrhabrraption discription

    Microsome - substrate - ingtrate system - 0.1m PBS (Ph7.4)

    • Qeb:
      Hauv cov khoom siv vitro metabolism
    • Yam khoom tsis tau.:
      0112B1.01
    • Chav Tsev Loj:
      0.2ml * 50 xeem
    • Cov ntaub so ntswg:
      Nplooj siab
    • Hom:
      Tus liab
    • Sib deev:
      Tus txiv neej
    • Kev Cia Cov Neeg Cia thiab Tsheb Thauj Mus Los:
      Khw ntawm - 70 ° C. Dej khov kom qhuav.
    • Yam tshuaj uas:
      Theem II metabolic Stability Kit (Umts)
    • Kuaj System:
      Microstre
    • Cov tau txais daim ntawv thov:
      Nyob rau hauv Versro kev ntsuas ntawm kev teeb meem ruaj khov

  • Yav dhau los:
  • Tom ntej:
  • Lus Xaiv