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IPHASE Phase II Metabolic Stability Kit,Monkey(Cynomolgus)

Tlhaloso e Khutšoanyane:

Phase II metabolism, eo hape e tsejoang e le karabelo e tlamang, e bua ka karabelo eo mohato oa I metabolites kapa lithethefatsi tsa prototype li kopanang le limolek'hule tse nyane tse sa feleng ka li-enzyme tsa mohato oa II, tse lebisang phokotsong ea chefo, ts'ebetso, kapa polarity ea lihlahisoa. Karolong ea II ea metabolism, karabelo e atileng haholo ke glucuronidation, eo ka nako eo uridine diphosphate glucuronic acid (UDPGA) e tlangoang ho prodrug ka catalyzation ka glucuronyl transferase ho li-microsomes. The glucuronide e eketsa ho qhibiliha ha metsi ho metabolites ho ntlafatsa mokelikeli. Sistimi ea metabolic ea phase II e ka hahuoa bocha ka motsoako oa li-microsomes tsa sebete le UGT mme ea sebelisoa ho ithuta botsitso ba karolo ea II ea bakuli ba lithethefatsi in vitro.

Lintlha tsa Sehlahisoa

Li-tag tsa Sehlahisoa

  • Tlhaloso ea lihlahisoa

    Microsome|Substrate| UGT Incubation System| 0.1M PBS (pH7.4)

    • Sehlopha:
      Lisebelisoa tsa in vitro metabolism
    • Ntho NO.:
      0112B1.02
    • Boholo ba Yuniti:
      0.2mL * 50 teko
    • Tishu:
      Sebete
    • Mefuta:
      Tshwene
    • Thobalano:
      E tšehali
    • Maemo a polokelo le lipalangoang:
      Boloka ho -70°C. Leqhoa le omileng le fanoa.
    • Mofuta oa tlhahlobo:
      Phase II Metabolic Stability Kit (UGTs)
    • Sistimi ea Teko:
      Microsome
    • Sebaka sa kopo:
      Tlhahlobo ea In vitro ea Botsitso ba Metabolic

  • E fetileng:
  • E latelang:
  • Khetho ea Puo