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IPHASE Phase II Metabolic Stability Kit, nas (ICR/CD-1)

Lus piav qhia luv luv:

Phase II metabolism, tseem hu ua kev sib khi cov tshuaj tiv thaiv, yog hais txog cov tshuaj tiv thaiv nyob rau theem I metabolites lossis cov tshuaj tiv thaiv ua ke nrog cov tshuaj endogenous me me los ntawm theem II enzymes, ua rau txo qis ntawm toxicity, kev ua, lossis polarity ntawm cov tshuaj. Hauv theem II metabolism, cov tshuaj tiv thaiv feem ntau yog glucuronidation, thaum lub sij hawm uridine diphosphate glucuronic acid (UDPGA) raug khi rau prodrug ntawm catalyzation los ntawm glucuronyl transferase hauv microsomes. Cov glucuronide tsim ua kom dej - solubility ntawm metabolites los txhim kho cov excretion. Phase II metabolic system tuaj yeem rov tsim dua los ntawm kev sib xyaw ntawm daim siab microsomes thiab UGT thiab siv los kawm theem II metabolic stability ntawm cov tshuaj sib tw hauv vitro.

Product Detail

Khoom cim npe

  • Cov khoom piav qhia

    Microsome |Substrate| UGT Incubation System| 0.1M PBS (pH7.4)

    • Qeb:
      Cov khoom siv hauv vitro metabolism
    • Yam khoom NO.:
      0112 E1.01
    • Unit Loj:
      0.2ml * 50 test
    • Cov ntaub so ntswg:
      Daim siab
    • Hom:
      Nas
    • Kev sib deev:
      Txiv neej
    • Cia tej yam kev mob thiab kev thauj mus los:
      Khaws ntawm - 70 ° C. Cov dej khov qhuav xa tuaj.
    • Hom kev xeem:
      Phase II Metabolic Stability Kit (UGTs)
    • Test System:
      Microsome
    • Scope ntawm kev siv:
      Nyob rau hauv vitro Kev ntsuam xyuas ntawm Metabolic Stability

  • Yav dhau los:
  • Tom ntej:
  • Xaiv hom lus