Adikole
Mukamachita kusanthula kwa pharmacokinetics, gawo lofunikira kwambiri pa cholumikizira cha mankhwala, adsorption, kugawa, kagayidwe kagayidwe, ndi mawu (adme) kuyenera kuyikiridwa mukamagwiritsa ntchito mankhwala. Ma metabolism, kapena biotransform, amatanthauza njira yomwe mankhwala omwe amagwiritsa ntchito mankhwala osokoneza bongo azomwe amayamwa ndikuthetsa thupi. Ogawidwa gawo la II & II kagayidwe, biotransform makamaka imapezeka m'chiwindi, chinthu chinacho chimalemedwa ndi michere ya metabolic, komanso m'matumbo, magazi, ndi khungu.
Njira yofunika kwambiri, yokhudza matenda a kagayidwe kambiri imachulukitsa kuti akhazikitse kukonzanso mankhwala a metabolic muumunthu, kugwiritsa ntchito mankhwala ndi chitetezo. Zaka zingapo zapitazi, Iphase yapanga zinthu zingapo zophunzitsira mankhwala osokoneza bongo kuphatikiza camezype, enzyme zoletsa (IC50). Kuphatikiza apo, Iphafa amaperekanso chothandiza mu - Mitundu ya Vitro monga hepatocytes, chiwindi ndi matumbo oyambira, cytosol, cytols, cytol, cytols, cytol, cytol, cytol, cytol, cytol, cytosol, cytol, cytol, cytol